@article{ChaikuadLangBrennanetal.2016, author = {Apirat Chaikuad and Steffen Lang and Paul E. Brennan and Claudia Temperini and Oleg Fedorov and Johan Hollander and Ruta Nachane and Chris Abell and Susanne M{\"u}ller and Gregg Siegal and Stefan Knapp}, title = {Structure-based identification of inhibitory fragments targeting the p300/CBP-associated factor bromodomain}, journal = {Journal of medicinal chemistry}, volume = {59}, number = {4}, pages = {1648 -- 1653}, doi = {10.1021/acs.jmedchem.5b01719}, year = {2016}, }