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1H, 13C, and 15N backbone chemical shift assignments of coronavirus-2 non-structural protein Nsp10
(2020)
Kubatova, Nina ; Qureshi, Nusrat ; Altınçekiç, Nadide ; Abele, Rupert ; Bains, Jasleen Kaur ; Ceylan, Betül ; Ferner, Jan ; Fuks, Christin ; Hargittay, Bruno ; Hutchison, Marie ; de Jesus, Vanessa ; Kutz, Felicitas ; Wirtz Martin, Maria Alexandra ; Meiser, Nathalie ; Linhard, Verena ; Pyper, Dennis Joshua ; Trucks, Sven ; Fürtig, Boris ; Hengesbach, Martin ; Löhr, Frank ; Richter, Christian ; Saxena, Krishna ; Schlundt, Andreas ; Schwalbe, Harald ; Sreeramulu, Sridhar ; Wacker, Anna ; Weigand, Julia ; Wirmer-Bartoschek, Julia ; Wöhnert, Jens
The international Covid19-NMR consortium aims at the comprehensive spectroscopic characterization of SARS-CoV-2 RNA elements and proteins and will provide NMR chemical shift assignments of the molecular components of this virus. The SARS-CoV-2 genome encodes approximately 30 different proteins. Four of these proteins are involved in forming the viral envelope or in the packaging of the RNA genome and are therefore called structural proteins. The other proteins fulfill a variety of functions during the viral life cycle and comprise the so-called non-structural proteins (nsps). Here, we report the near-complete NMR resonance assignment for the backbone chemical shifts of the non-structural protein 10 (nsp10). Nsp10 is part of the viral replication-transcription complex (RTC). It aids in synthesizing and modifying the genomic and subgenomic RNAs. Via its interaction with nsp14, it ensures transcriptional fidelity of the RNA-dependent RNA polymerase, and through its stimulation of the methyltransferase activity of nsp16, it aids in synthesizing the RNA cap structures which protect the viral RNAs from being recognized by the innate immune system. Both of these functions can be potentially targeted by drugs. Our data will aid in performing additional NMR-based characterizations, and provide a basis for the identification of possible small molecule ligands interfering with nsp10 exerting its essential role in viral replication.
Martin-Subero, Jose Ignacio ; Ammerpohl, Ole ; Bibikova, Marina ; Wickham-Garcia, Eliza ; Agirre, Xabier ; Alvarez, Sara ; Brüggemann, Monika ; Bug, Stefanie ; Calasanz, Maria J. ; Deckert, Martina ; Dreyling, Martin ; Du, Ming Q. ; Dürig, Jan ; Dyer, Martin J. S. ; Fan, Jian-Bing ; Gesk, Stefan ; Hansmann, Martin-Leo ; Harder, Lana ; Hartmann, Sylvia ; Klapper, Wolfram ; Küppers, Ralf ; Montesinos-Rongen, Manuel ; Nagel, Inga ; Pott, Christiane ; Richter, Julia ; Román-Gómez, José ; Seifert, Marc ; Stein, Harald ; Suela, Javier ; Trümper, Lorenz ; Vater, Inga ; Prosper, Felipe ; Haferlach, Claudia ; Cruz Cigudosa, Juan ; Siebert, Reiner
Background: Alterations in the DNA methylation pattern are a hallmark of leukemias and lymphomas. However, most epigenetic studies in hematologic neoplasms (HNs) have focused either on the analysis of few candidate genes or many genes and few HN entities, and comprehensive studies are required. Methodology/Principal Findings: Here, we report for the first time a microarray-based DNA methylation study of 767 genes in 367 HNs diagnosed with 16 of the most representative B-cell (n = 203), T-cell (n = 30), and myeloid (n = 134) neoplasias, as well as 37 samples from different cell types of the hematopoietic system. Using appropriate controls of B-, T-, or myeloid cellular origin, we identified a total of 220 genes hypermethylated in at least one HN entity. In general, promoter hypermethylation was more frequent in lymphoid malignancies than in myeloid malignancies, being germinal center mature B-cell lymphomas as well as B and T precursor lymphoid neoplasias those entities with highest frequency of gene-associated DNA hypermethylation. We also observed a significant correlation between the number of hypermethylated and hypomethylated genes in several mature B-cell neoplasias, but not in precursor B- and T-cell leukemias. Most of the genes becoming hypermethylated contained promoters with high CpG content, and a significant fraction of them are targets of the polycomb repressor complex. Interestingly, T-cell prolymphocytic leukemias show low levels of DNA hypermethylation and a comparatively large number of hypomethylated genes, many of them showing an increased gene expression. Conclusions/Significance: We have characterized the DNA methylation profile of a wide range of different HNs entities. As well as identifying genes showing aberrant DNA methylation in certain HN subtypes, we also detected six genes—DBC1, DIO3, FZD9, HS3ST2, MOS, and MYOD1—that were significantly hypermethylated in B-cell, T-cell, and myeloid malignancies. These might therefore play an important role in the development of different HNs.