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Adamczyk, Leszek ; Agakishiev, Geydar ; Aggarwal, Madan Mohan ; Ahammed, Zubayer ; Alakhverdyants, A. V. ; Alekseev, Igor G. ; Alford, J. ; Anderson, Bryon D. ; Anson, Christopher Daniel ; Arkhipkin, Dmitry A. ; Averichev, Georgy S. ; Balewski, Jan ; Banerjee, A. ; Barnovska, Z. ; Beavis, D. R. ; Bellwied, Rene ; Betancourt, M. J. ; Betts, R. R. ; Bhasin, Anju ; Bhati, Ashok Kumar ; Bichsel, Hans ; Bielčík, Jaroslav ; Bielčíková, Jana ; Bland, Leslie C. ; Bordyuzhin, Igor G. ; Borowski, W. ; Bouchet, J. ; Brandin, Andrei V. ; Brovko, S. G. ; Bruna, Elena ; Bueltmann, S. ; Bunzarov, Ivan ; Burton, T. P. ; Butterworth, Joseph ; Cai, Xiang-Zhou ; Caines, Helen Louise ; Calderón de la Barca Sánchez, Manuel ; Cebra, Daniel A. ; Cendejas, R. ; Cervantes, M. C. ; Chaloupka, Petr ; Chattopadhyay, S. ; Chen, H. F. ; Chen, J. H. ; Chen, J. Y. ; Chen, L. ; Cheng, J. ; Cherney, Michael Gerard ; Chikanian, Alexei ; Christie, William ; Chung, P. ; Chwastowski, J. ; Codrington, M. J. M. ; Corliss, R. ; Cramer, John G. ; Crawford, Henry J. ; Cui, X. ; Davila Leyva, A. ; De Silva, L. C. ; Debbe, R. R. ; Dedovich, T. G. ; Deng, J. ; Souza, Rafael Derradi de ; Dhamija, S. ; Didenko, Lidia ; Ding, F. ; Djawotho, P. ; Dong, X. ; Drachenberg, James Lucus ; Draper, James E. ; Du, C. M. ; Dunkelberger, L. E. ; Dunlop, James C. ; Efimov, Leonid G. ; Elnimr, M. ; Engelage, Jon M. ; Eppley, Geary Wareham ; Eun, L. ; Evdokimov, Olga Y. ; Fatemi, Renee H. ; Fedorišin, Jan ; Fersch, R. G. ; Filip, Peter ; Finch, Evan ; Fisyak, Yuri V. ; Gagliardi, Carl A. ; Gangadharan, Dhevan Raja ; Geurts, Frank ; Gliske, S. ; Gorbunov, Y. N. ; Grebenyuk, O. G. ; Grosnick, David P. ; Gupta, S. ; Guryn, Włodzimierz ; Haag, B. ; Hajkova, O. ; Hamed, Ahmed M. ; Han, L-X. ; Harris, John W. ; Hays-Wehle, J. P. ; Heppelmann, S. ; Hirsch, Andrew S. ; Hoffmann, Gerald W. ; Hofman, D. J. ; Horvat, S. ; Huang, Bingchu ; Huang, Huan Zhong ; Huck, P. ; Humanic, Thomas J. ; Huo, L. ; Igo, George J. ; Jacobs, William W. ; Jena, Chitrasen ; Joseph, J. ; Judd, Eleanor G. ; Kabana, Sonia ; Kang, K. ; Kapitan, J. ; Kauder, Kolja ; Ke, Hongwei ; Keane, Declan ; Kechechyan, Armen ; Kesich, A. ; Kettler, D. ; Kikola, D. P. ; Kiryluk, Joanna ; Kisiel, Adam Ryszard ; Kizka, V. ; Klein, Spencer Robert ; Koetke, Donald D. ; Kollegger, Thorsten ; Konzer, J. ; Koralt, I. ; Koroleva, L. ; Korsch, W. ; Kotchenda, L. ; Kravtsov, Peter ; Krueger, Keith William ; Kumar, Lokesh ; Lamont, Matthew A. C. ; Landgraf, Jeffery M. ; LaPointe, S. ; Lauret, Jerome ; Lebedev, Alexei ; Lednicky, Richard ; Lee, J. H. ; Leight, W. ; LeVine, Micheal J. ; Li, C. ; Li, L. ; Li, W. ; Li, X. ; Li, X. ; Li, Y. ; Li, Z. M. ; Lima, L. M. ; Lisa, Michael A. ; Liu, F. ; Ljubicic, Tonko A. ; Llope, William Joseph ; Longacre, Ronald S. ; Lu, Y. ; Luo, X. ; Luszczak, A. ; Ma, G. L. ; Ma, Yu-Gang ; Mahapatra, Durga Prasad ; Majka, Richard Daniel ; Mall, O. I. ; Margetis, Spyridon ; Markert, Christina ; Masui, H. ; Matis, Howard S. ; McDonald, Daniel ; McShane, Tom S. ; Mioduszewski, Saskia ; Mitrovski, M. K. ; Mohammed, Y. ; Mohanty, Bedangadas ; Morozov, B. ; Munhoz, Marcelo Gameiro ; Mustafa, M. K. ; Naglis, M. ; Nandi, Basanta Kumar ; Nasim, Md. ; Nayak, Tapan Kumar ; Nogach, Larisa V. ; Odyniec, Grazyna Janina ; Ogawa, Akio ; Oh, K. ; Ohlson, Alice ; Okorokov, Vitaly A. ; Oldag, E. W. ; Oliveira, R. A. N. ; Olson, Douglas L. ; Pachr, Miloš ; Page, Brian S. ; Pal, Susanta Kumar ; Pan, Y. X. ; Pandit, Y. ; Panebratsev, Yuri ; Pawlak, Tomasz Jan ; Pawlik, Bogdan ; Pei, Hua ; Perkins, Chris ; Peryt, Wiktor Stanislaw ; Pile, P. ; Planinic, Mirko ; Pluta, Jan Marian ; Plyku, D. ; Poljak, Nikola ; Porter, Jeffrey Brent ; Poskanzer, Arthur M. ; Powell, C. B. ; Prindle, Duncan J. ; Pruneau, Claude A. ; Pruthi, Navneet Kumar ; Przybycien, Mariusz ; Pujahari, P. R. ; Putschke, Jörn H. ; Qiu, H. ; Raniwala, Rashmi ; Raniwala, Sudhir ; Ray, Robert L. ; Redwine, R. ; Reed, Rosi Jan ; Riley, C. K. ; Ritter, Hans Georg ; Roberts, Jabus B. ; Rogačevskij, Oleg V. ; Romero, Juan L. ; Ruan, L. ; Rusnak, Jan ; Sahoo, Nihar Ranjan ; Sakrejda, Iwona ; Salur, Sevil ; Sandweiss, Jack H. ; Sangaline, E. ; Sarkar, Amal ; Schambach, Joachim ; Scharenberg, Rolf Paul ; Schmah, A. M. ; Schmitz, Norbert ; Schuster, T. R. ; Seele, J. ; Seger, Janet Elizabeth ; Seyboth, Peter ; Shah, N. ; Shahaliev, Ehtiram ; Shao, M. ; Sharma, B. ; Sharma, M. ; Shi, Shusu ; Shou, Q. Y. ; Sichtermann, Ernst P. ; Singaraju, Rama Narayana ; Skoby, Michael J. ; Smirnov, Nikolai ; Solanki, D. ; Sorensen, Paul Richard ; deSouza, U. G. ; Spinka, Harold. M. ; Srivastava, B. ; Stanislaus, T. D. Shirvel ; Steadman, S. G. ; Stevens, J. R. ; Stock, Reinhard ; Strichanov, Michail Nikolaevič ; Stringfellow, Blair ; Suaide, Alexandre Alarcon do Passo ; Suarez, M. C. ; Šumbera, Michal ; Sun, X. M. ; Sun, Y. ; Sun, Z. ; Surrow, Bernd ; Svirida, Dmitry N. ; Symons, Timothy James MacNeil ; Toledo, Alejandro Szanto de ; Takahashi, Jun ; Tang, Aihong ; Tang, Zebo ; Tarini, L. H. ; Tarnowsky, Terence J. ; Thein, Dylan ; Thomas, James H. ; Tian, J. ; Timmins, Anthony Robert ; Tlusty, David ; Tokarev, Mikhail V. ; Trainor, Thomas A. ; Trentalange, Stephen ; Tribble, Robert E. ; Tribedy, Prithwish ; Trzeciak, Barbara Antonina ; Tsai, Oleg D. ; Turnau, J. ; Ullrich, Thomas ; Underwood, David G. ; Van Buren, Gene ; van Nieuwenhuizen, G. ; Vanfossen, J. A. ; Varma, Raghava ; Vasconcelos, G. M. S. ; Videbæk, Flemming ; Viyogi, Yogendra P. ; Vokal, Stanislav ; Voloshin, Sergei ; Vossen, A. ; Wada, M. ; Wang, F. ; Wang, G. ; Wang, H. ; Wang, J. S. ; Wang, Q. ; Wang, X. L. ; Wang, Y. ; Webb, Grant ; Webb, Jason C. ; Westfall, Gary D. ; Whitten, Charles A. ; Wieman, Howard ; Wissink, Scott W. ; Witt, Richard ; Witzke, W. ; Wu, Y. F. ; Xiao, Z. ; Xie, W. ; Xin, K. ; Xu, H. ; Xu, N. ; Xu, Qinghua ; Xu, W. ; Xu, Y. ; Xu, Z. ; Xue, L. ; Yang, Y. ; Yang, Y. ; Yepes, Pablo P. ; Yi, Y. ; Yip, K. ; Yoo, I-K. ; Zawisza, M. ; Zbroszczyk, Hanna Paulina ; Zhang, J. B. ; Zhang, S. ; Zhang, W. M. ; Zhang, X. P. ; Zhang, Y. ; Zhang, Z. P. ; Zhao, F. ; Zhao, J. ; Zhong, C. ; Zhu, X. ; Zhu, Y. H. ; Zoulkarneeva, Youlia
STAR's measurements of directed flow (v1) around midrapidity for π±, K±, K0S, p and p¯ in Au + Au collisions at $\sqrtsNN = 200$ GeV are presented. A negative v1(y) slope is observed for most of produced particles (π±, K±, K0S and p¯). The proton v1(y) slope is found to be much closer to zero compared to antiprotons. A sizable difference is seen between v1 of protons and antiprotons in 5-30% central collisions. The v1 excitation function is presented. Comparisons to model calculations (RQMD, UrQMD, AMPT, QGSM with parton recombination, and a hydrodynamics model with a tilted source) are made. Anti-flow alone cannot explain the centrality dependence of the difference between the v1(y) slopes of protons and antiprotons.
Adamczyk, Leszek ; Agakishiev, Geydar ; Aggarwal, Madan Mohan ; Ahammed, Zubayer ; Alakhverdyants, A. V. ; Alekseev, Igor G. ; Alford, J. ; Anderson, Bryon D. ; Anson, Christopher Daniel ; Arkhipkin, Dmitry A. ; Averichev, Georgy S. ; Balewski, Jan ; Banerjee, A. ; Barnovska, Z. ; Beavis, D. R. ; Bellwied, Rene ; Betancourt, M. J. ; Betts, R. R. ; Bhasin, Anju ; Bhati, Ashok Kumar ; Bichsel, Hans ; Bielčík, Jaroslav ; Bielčíková, Jana ; Bland, Leslie C. ; Bordyuzhin, Igor G. ; Borowski, W. ; Bouchet, J. ; Brandin, Andrei V. ; Brovko, S. G. ; Bruna, Elena ; Bueltmann, S. ; Bunzarov, Ivan ; Burton, T. P. ; Butterworth, Joseph ; Cai, Xiang-Zhou ; Caines, Helen Louise ; Calderón de la Barca Sánchez, Manuel ; Cebra, Daniel A. ; Cendejas, R. ; Cervantes, M. C. ; Chaloupka, Petr ; Chattopadhyay, S. ; Chen, H. F. ; Chen, J. H. ; Chen, J. Y. ; Chen, L. ; Cheng, J. ; Cherney, Michael Gerard ; Chikanian, Alexei ; Christie, William ; Chung, P. ; Chwastowski, J. ; Codrington, M. J. M. ; Corliss, R. ; Cramer, John G. ; Crawford, Henry J. ; Cui, X. ; Davila Leyva, A. ; De Silva, L. C. ; Debbe, R. R. ; Dedovich, T. G. ; Deng, J. ; Souza, Rafael Derradi de ; Dhamija, S. ; Didenko, Lidia ; Ding, F. ; Djawotho, P. ; Dong, X. ; Drachenberg, James Lucus ; Draper, James E. ; Du, C. M. ; Dunkelberger, L. E. ; Dunlop, James C. ; Efimov, Leonid G. ; Elnimr, M. ; Engelage, Jon M. ; Eppley, Geary Wareham ; Eun, L. ; Evdokimov, Olga Y. ; Fatemi, Renee H. ; Fedorišin, Jan ; Fersch, R. G. ; Filip, Peter ; Finch, Evan ; Fisyak, Yuri V. ; Gagliardi, Carl A. ; Gangadharan, Dhevan Raja ; Geurts, Frank ; Gliske, S. ; Gorbunov, Y. N. ; Grebenyuk, O. G. ; Grosnick, David P. ; Gupta, S. ; Guryn, Włodzimierz ; Haag, B. ; Hajkova, O. ; Hamed, Ahmed M. ; Han, L-X. ; Harris, John W. ; Hays-Wehle, J. P. ; Heppelmann, S. ; Hirsch, Andrew S. ; Hoffmann, Gerald W. ; Hofman, D. J. ; Horvat, S. ; Huang, Bingchu ; Huang, Huan Zhong ; Huck, P. ; Humanic, Thomas J. ; Huo, L. ; Igo, George J. ; Jacobs, William W. ; Jena, Chitrasen ; Joseph, J. ; Judd, Eleanor G. ; Kabana, Sonia ; Kang, K. ; Kapitan, J. ; Kauder, Kolja ; Ke, Hongwei ; Keane, Declan ; Kechechyan, Armen ; Kesich, A. ; Kettler, D. ; Kikola, D. P. ; Kiryluk, Joanna ; Kisiel, Adam Ryszard ; Kizka, V. ; Klein, Spencer Robert ; Koetke, Donald D. ; Kollegger, Thorsten ; Konzer, J. ; Koralt, I. ; Koroleva, L. ; Korsch, W. ; Kotchenda, L. ; Kravtsov, Peter ; Krueger, Keith William ; Kumar, Lokesh ; Lamont, Matthew A. C. ; Landgraf, Jeffery M. ; LaPointe, S. ; Lauret, Jerome ; Lebedev, Alexei ; Lednicky, Richard ; Lee, J. H. ; Leight, W. ; LeVine, Micheal J. ; Li, C. ; Li, L. ; Li, W. ; Li, X. ; Li, X. ; Li, Y. ; Li, Z. M. ; Lima, L. M. ; Lisa, Michael A. ; Liu, F. ; Ljubicic, Tonko A. ; Llope, William Joseph ; Longacre, Ronald S. ; Lu, Y. ; Luo, X. ; Luszczak, A. ; Ma, G. L. ; Ma, Yu-Gang ; Mahapatra, Durga Prasad ; Majka, Richard Daniel ; Mall, O. I. ; Margetis, Spyridon ; Markert, Christina ; Masui, H. ; Matis, Howard S. ; McDonald, Daniel ; McShane, Tom S. ; Mioduszewski, Saskia ; Mitrovski, M. K. ; Mohammed, Y. ; Mohanty, Bedangadas ; Morozov, B. ; Munhoz, Marcelo Gameiro ; Mustafa, M. K. ; Naglis, M. ; Nandi, Basanta Kumar ; Nasim, Md. ; Nayak, Tapan Kumar ; Nogach, Larisa V. ; Odyniec, Grazyna Janina ; Ogawa, Akio ; Oh, K. ; Ohlson, Alice ; Okorokov, Vitaly A. ; Oldag, E. W. ; Oliveira, R. A. N. ; Olson, Douglas L. ; Pachr, Miloš ; Page, Brian S. ; Pal, Susanta Kumar ; Pan, Y. X. ; Pandit, Y. ; Panebratsev, Yuri ; Pawlak, Tomasz Jan ; Pawlik, Bogdan ; Pei, Hua ; Perkins, Chris ; Peryt, Wiktor Stanislaw ; Pile, P. ; Planinic, Mirko ; Pluta, Jan Marian ; Plyku, D. ; Poljak, Nikola ; Porter, Jeffrey Brent ; Poskanzer, Arthur M. ; Powell, C. B. ; Prindle, Duncan J. ; Pruneau, Claude A. ; Pruthi, Navneet Kumar ; Przybycien, Mariusz ; Pujahari, P. R. ; Putschke, Jörn H. ; Qiu, H. ; Raniwala, Rashmi ; Raniwala, Sudhir ; Ray, Robert L. ; Redwine, R. ; Reed, Rosi Jan ; Riley, C. K. ; Ritter, Hans Georg ; Roberts, Jabus B. ; Rogačevskij, Oleg V. ; Romero, Juan L. ; Ruan, L. ; Rusnak, Jan ; Sahoo, Nihar Ranjan ; Sakrejda, Iwona ; Salur, Sevil ; Sandweiss, Jack H. ; Sangaline, E. ; Sarkar, Amal ; Schambach, Joachim ; Scharenberg, Rolf Paul ; Schmah, A. M. ; Schmitz, Norbert ; Schuster, T. R. ; Seele, J. ; Seger, Janet Elizabeth ; Seyboth, Peter ; Shah, N. ; Shahaliev, Ehtiram ; Shao, M. ; Sharma, B. ; Sharma, M. ; Shi, Shusu ; Shou, Q. Y. ; Sichtermann, Ernst P. ; Singaraju, Rama Narayana ; Skoby, Michael J. ; Smirnov, Nikolai ; Solanki, D. ; Sorensen, Paul Richard ; deSouza, U. G. ; Spinka, Harold. M. ; Srivastava, B. ; Stanislaus, T. D. Shirvel ; Steadman, S. G. ; Stevens, J. R. ; Stock, Reinhard ; Strichanov, Michail Nikolaevič ; Stringfellow, Blair ; Suaide, Alexandre Alarcon do Passo ; Suarez, M. C. ; Šumbera, Michal ; Sun, X. M. ; Sun, Y. ; Sun, Z. ; Surrow, Bernd ; Svirida, Dmitry N. ; Symons, Timothy James MacNeil ; Toledo, Alejandro Szanto de ; Takahashi, Jun ; Tang, Aihong ; Tang, Zebo ; Tarini, L. H. ; Tarnowsky, Terence J. ; Thein, Dylan ; Thomas, James H. ; Tian, J. ; Timmins, Anthony Robert ; Tlusty, David ; Tokarev, Mikhail V. ; Trainor, Thomas A. ; Trentalange, Stephen ; Tribble, Robert E. ; Tribedy, Prithwish ; Trzeciak, Barbara Antonina ; Tsai, Oleg D. ; Turnau, J. ; Ullrich, Thomas ; Underwood, David G. ; Van Buren, Gene ; van Nieuwenhuizen, G. ; Vanfossen, J. A. ; Varma, Raghava ; Vasconcelos, G. M. S. ; Videbæk, Flemming ; Viyogi, Yogendra P. ; Vokal, Stanislav ; Voloshin, Sergei ; Vossen, A. ; Wada, M. ; Wang, F. ; Wang, G. ; Wang, H. ; Wang, J. S. ; Wang, Q. ; Wang, X. L. ; Wang, Y. ; Webb, Grant ; Webb, Jason C. ; Westfall, Gary D. ; Whitten, Charles A. ; Wieman, Howard ; Wissink, Scott W. ; Witt, Richard ; Witzke, W. ; Wu, Y. F. ; Xiao, Z. ; Xie, W. ; Xin, K. ; Xu, H. ; Xu, N. ; Xu, Qinghua ; Xu, W. ; Xu, Y. ; Xu, Z. ; Xue, L. ; Yang, Y. ; Yang, Y. ; Yepes, Pablo P. ; Yi, Y. ; Yip, K. ; Yoo, I-K. ; Zawisza, M. ; Zbroszczyk, Hanna Paulina ; Zhang, J. B. ; Zhang, S. ; Zhang, W. M. ; Zhang, X. P. ; Zhang, Y. ; Zhang, Z. P. ; Zhao, F. ; Zhao, J. ; Zhong, C. ; Zhu, X. ; Zhu, Y. H. ; Zoulkarneeva, Youlia
STAR's measurements of directed flow (v1) around midrapidity for π±, K±, K0S, p and p¯ in Au + Au collisions at $\sqrtsNN = 200$ GeV are presented. A negative v1(y) slope is observed for most of produced particles (π±, K±, K0S and p¯). In 5-30% central collisions a sizable difference is present between the v1(y) slope of protons and antiprotons, with the former being consistent with zero within errors. The v1 excitation function is presented. Comparisons to model calculations (RQMD, UrQMD, AMPT, QGSM with parton recombination, and a hydrodynamics model with a tilted source) are made. For those models which have calculations of v1 for both pions and protons, none of them can describe v1(y) for pions and protons simultaneously. The hydrodynamics model with a tilted source as currently implemented cannot explain the centrality dependence of the difference between the v1(y) slopes of protons and antiprotons.
Unique features of a global human ectoparasite identified through sequencing of the bed bug genome
(2016)
Benoit, Joshua B. ; Adelman, Zach N. ; Reinhardt, Klaus ; Dolan, Amanda ; Poelchau, Monica ; Jennings, Emily C. ; Szuter, Elise M. ; Hagan, Richard W. ; Gujar, Hemant ; Shukla, Jayendra Nath ; Zhu, Fang ; Mohan, Muthugounder ; Nelson, David R. ; Rosendale, Andrew J. ; Derst, Christian ; Resnik, Valentina ; Wernig, Sebastian ; Menegazzi, Pamela ; Wegener, Christian ; Peschel, Nicolai ; Hendershot, Jacob M. ; Blenau, Wolfgang ; Predel, Reinhard ; Johnston, Paul R. ; Ioannidis, Panagiotis ; Waterhouse, Robert M. ; Nauen, Ralf ; Schorn, Corinna ; Ott, Mark-Christoph ; Maiwald, Frank ; Johnston, J. Spencer ; Gondhalekar, Ameya D. ; Scharf, Michael E. ; Peterson, Brittany F. ; Raje, Kapil R. ; Hottel, Benjamin A. ; Armisén, David ; Crumière, Antonin Jean Johan ; Refki, Peter Nagui ; Santos, Maria Emilia ; Sghaier, Essia ; Viala, Séverine ; Khila, Abderrahman ; Ahn, Seung-Joon ; Childers, Christopher ; Lee, Chien-Yueh ; Lin, Han ; Hughes, Daniel S. T. ; Duncan, Elizabeth J. ; Murali, Shwetha C. ; Qu, Jiaxin ; Dugan, Shannon ; Lee, Sandra L. ; Chao, Hsu ; Dinh, Huyen ; Han, Yi ; Doddapaneni, Harshavardhan ; Worley, Kim C. ; Muzny, Donna Marie ; Wheeler, David ; Panfilio, Kristen A. ; Vargas Jentzsch, Iris M. ; Vargo, Edward L. ; Booth, Warren ; Friedrich, Markus ; Weirauch, Matthew T. ; Anderson, Michelle A. ; Jones, Jeffery W. ; Mittapalli, Omprakash ; Zhao, Chaoyang ; Zhou, Jing-Jiang ; Evans, Jay D. ; Attardo, Geoffrey M. ; Robertson, Hugh M. ; Zdobnov, Evgeny M. ; Ribeiro, José M. C. ; Gibbs, Richard A. ; Werren, John H. ; Palli, Subba Reddy ; Schal, Coby ; Richards, Stephen
The bed bug, Cimex lectularius, has re-established itself as a ubiquitous human ectoparasite throughout much of the world during the past two decades. This global resurgence is likely linked to increased international travel and commerce in addition to widespread insecticide resistance. Analyses of the C. lectularius sequenced genome (650 Mb) and 14,220 predicted protein-coding genes provide a comprehensive representation of genes that are linked to traumatic insemination, a reduced chemosensory repertoire of genes related to obligate hematophagy, host–symbiont interactions, and several mechanisms of insecticide resistance. In addition, we document the presence of multiple putative lateral gene transfer events. Genome sequencing and annotation establish a solid foundation for future research on mechanisms of insecticide resistance, human–bed bug and symbiont–bed bug associations, and unique features of bed bug biology that contribute to the unprecedented success of C. lectularius as a human ectoparasite.
Bauer, Matthias R. ; Jones, Rhiannon N. ; Baud, Matthias G. J. ; Wilcken, Rainer ; Böckler, Frank ; Fersht, Alan ; Jörger, Andreas C. ; Spencer, John
Many oncogenic mutants of the tumor suppressor p53 are conformationally unstable, including the frequently occurring Y220C mutant. We have previously developed several small-molecule stabilizers of this mutant. One of these molecules, PhiKan083, 1-(9-ethyl-9H-carbazole-3-yl)-N-methylmethanamine, binds to a mutation-induced surface crevice with a KD = 150 μM, thereby increasing the melting temperature of the protein and slowing its rate of aggregation. Incorporation of fluorine atoms into small molecule ligands can substantially improve binding affinity to their protein targets. We have, therefore, harnessed fluorine–protein interactions to improve the affinity of this ligand. Step-wise introduction of fluorines at the carbazole ethyl anchor, which is deeply buried within the binding site in the Y220C–PhiKan083 complex, led to a 5-fold increase in affinity for a 2,2,2-trifluoroethyl anchor (ligand efficiency of 0.3 kcal mol–1 atom–1). High-resolution crystal structures of the Y220C–ligand complexes combined with quantum chemical calculations revealed favorable interactions of the fluorines with protein backbone carbonyl groups (Leu145 and Trp146) and the sulfur of Cys220 at the mutation site. Affinity gains were, however, only achieved upon trifluorination, despite favorable interactions of the mono- and difluorinated anchors with the binding pocket, indicating a trade-off between energetically favorable protein–fluorine interactions and increased desolvation penalties. Taken together, the optimized carbazole scaffold provides a promising starting point for the development of high-affinity ligands to reactivate the tumor suppressor function of the p53 mutant Y220C in cancer cells.
Effect of event selection on jetlike correlation measurement in d+Au collisions at √sNN = 200 GeV
(2015)
Adamczyk, Leszek ; Adkins, J. Kevin ; Agakishiev, Geydar ; Aggarwal, Madan Mohan ; Ahammed, Zubayer ; Alekseev, Igor G. ; Alford, J. ; Aparin, Alexey ; Arkhipkin, Dmitry A. ; Aschenauer, Elke Caroline ; Averichev, Georgy S. ; Banerjee, A. ; Bellwied, Rene ; Bhasin, Anju ; Bhati, Ashok Kumar ; Bhattarai, P. ; Bielčík, Jaroslav ; Bielčíková, Jana ; Bland, Leslie C. ; Bordyuzhin, Igor G. ; Bouchet, Jonathan ; Brandin, Andrei V. ; Bunzarov, Ivan ; Burton, T.P. ; Butterworth, Joseph ; Caines, Helen Louise ; Calderón de la Barca Sánchez, Manuel ; Campbell, J.M. ; Cebra, Daniel A. ; Cervantes, M.C. ; Chakaberia, Irakli ; Chaloupka, Petr ; Chang, Z. ; Chattopadhyay, S. ; Chen, J.H. ; Cheng, J. ; Cherney, Michael Gerard ; Christie, William ; Codrington, M.J.M. ; Contin, Giacomo ; Crawford, Henry J. ; Das, Supriya ; De Silva, L.C. ; Debbe, R.R. ; Dedovič, Tatiana G. ; Deng, J. ; Derevschikov, Anatoly A. ; Souza, Rafael Derradi de ; di Ruzza, Benedetto ; Didenko, Lidia ; Dilks, Christopher ; Dong, X. ; Drachenberg, James Lucus ; Draper, James E. ; Du, C.M. ; Dunkelberger, Lloyd Edward ; Dunlop, James C. ; Efimov, Leonid G. ; Engelage, Jon M. ; Eppley, Geary Wareham ; Esha, Roli ; Evdokimov, Olga Y. ; Eyser, Kjeld Oleg ; Fatemi, Renee H. ; Fazio, Salvatore ; Federič, Pavol ; Fedorišin, Jan ; Feng ; Filip, Peter ; Fisyak, Yuri V. ; Flores, C.E. ; Gagliardi, Carl A. ; Garand, David ; Geurts, Frank ; Gibson, Adam ; Girard, M. ; Greiner, Leo Clifford ; Grosnick, David P. ; Gunarathne, D.S. ; Guo, Y. ; Gupta, S. ; Gupta, Anik ; Guryn, Włodzimierz ; Hamad, Ayman ; Hamed, Ahmed M. ; Haque, R. ; Harris, John W. ; He, L. ; Heppelmann, Steven Francis ; Hirsch, Andrew S. ; Hoffmann, Gerald W. ; Hofman, D.J. ; Horvat, S. ; Huang, H.Z. ; Huang, X. ; Huang, B. ; Huck, Patrick ; Humanic, Thomas J. ; Igo, George J. ; Jacobs, William W. ; Jang, H. ; Judd, Eleanor G. ; Kabana, Sonia ; Kalinkin, Dmitry ; Kang, K. ; Kauder, Kolja ; Ke, Hongwei ; Keane, Declan ; Kechechyan, Armen ; Khan, Z.H. ; Kikola, D.P. ; Kisel, Ivan ; Kisiel, Adam Ryszard ; Klein, Spencer Robert ; Koetke, Donald D. ; Kollegger, Thorsten ; Kosarzewski, Leszek Krzysztof ; Kotchenda, L. ; Kraishan, A.F. ; Kravtsov, Peter ; Krueger, Keith William ; Kulakov, Igor ; Kumar, Lokesh ; Kycia, R.A. ; Lamont, Matthew A. C. ; Landgraf, Jeffery M. ; Landry, K.D. ; Lauret, Jerome ; Lebedev, Alexei ; Lednicky, Richard ; Lee, J.H. ; Li, Xiaomei ; Li, C. ; Li, Xiaomei ; Li, W. ; Li, Z.M. ; Li, Y. ; Lisa, Michael A. ; Liu, F. ; Ljubicic, Tonko A. ; Llope, William Joseph ; Lomnitz, Michael ; Longacre, Ronald S. ; Luo, X. ; Ma, L. ; Ma, G.L. ; Ma, Yu-Gang ; Ma, R. ; Magdy Abdelwahab Abdelrahman, Niseem ; Majka, Richard Daniel ; Manion, A. ; Margetis, Spyridon ; Markert, Christina ; Masui, H. ; Matis, Howard S. ; McDonald, Daniel ; Minaev, Nikolai G. ; Mioduszewski, Saskia ; Mohanty, Bedangadas ; Mondal, Mriganka Mouli ; Morozov, Dmitry A. ; Mustafa, M.K. ; Nandi, Basanta Kumar ; Nasim, Md. ; Nayak, Tapan Kumar ; Nigmatkulov, Grigory A. ; Nogach, Larisa V. ; Noh, S.Y. ; Novak, J. ; Nurušev, Sandibek B. ; Odyniec, Grazyna Janina ; Ogawa, Akio ; Oh, Kunsu ; Okorokov, Vitaly A. ; Olvitt, D.L. ; Page, Brian S. ; Pan, Y.X. ; Pandit, Y. ; Panebratsev, Yuri ; Pawlak, Tomasz Jan ; Pawlik, Bogdan ; Pei, Hua ; Perkins, Chris ; Pile, P. ; Planinic, Mirko ; Pluta, Jan Marian ; Poljak, Nikola ; Poniatowska, K. ; Porter, Jeffrey Brent ; Poskanzer, Arthur M. ; Pruthi, Navneet Kumar ; Przybycien, Mariusz ; Putschke, Jörn H. ; Qiu, H. ; Quintero, Amilkar ; Ramachandran, Suvarna ; Raniwala, Rashmi ; Raniwala, Sudhir ; Ray, Robert L. ; Ritter, Hans Georg ; Roberts, Jabus B. ; Rogačevskij, Oleg V. ; Romero, Juan L. ; Roy, Ankhi ; Ruan, Lijuan ; Rusnak, Jan ; Rusnakova, Olga ; Sahoo, Nihar Ranjan ; Sahu, Pradip Kumar ; Sakrejda, Iwona ; Salur, Sevil ; Sandacz, Andrzej ; Sandweiss, Jack H. ; Sarkar, Amal ; Schambach, Joachim ; Scharenberg, Rolf Paul ; Schmah, Alexander ; Schmidke, William B. ; Schmitz, Norbert ; Seger, Janet Elizabeth ; Seyboth, Peter ; Shah, N. ; Shahaliev, Ehtiram ; Shanmuganathan, Prashanth V. ; Shao, M. ; Sharma, B. ; Sharma, M.K. ; Shen, W.Q. ; Shi, S.S. ; Shou, Q.Y. ; Sichtermann, Ernst P. ; Šimko, Miroslav ; Skoby, M.J. ; Smirnov, Dmitri V. ; Smirnov, Nikolai ; Solanki, D. ; Song, L. ; Sorensen, Paul Richard ; Spinka, Harold. M. ; Srivastava, Brijesh Kumar ; Stanislaus, T. D. Shirvel ; Stock, Reinhard ; Strichanov, Michail Nikolaevič ; Stringfellow, Blair ; Šumbera, Michal ; Summa, B.J. ; Sun, Z. ; Sun, Y. ; Sun, X. ; Sun, X.M. ; Surrow, Bernd ; Svirida, Dmitry N. ; Szelezniak, M.A. ; Takahashi, Jun ; Tang, Zebo ; Tang, Aihong ; Tarnowsky, Terence J. ; Tawfik, Abdel Nasser ; Thomas, James H. ; Timmins, Anthony Robert ; Tlusty, David ; Tokarev, Mikhail V. ; Trentalange, Stephen ; Tribble, Robert E. ; Tribedy, Prithwish ; Tripathy, Srikanta Kumar ; Trzeciak, Barbara Antonina ; Tsai, Oleg D. ; Turnau, J. ; Ullrich, Thomas ; Underwood, David G. ; Upsal, Isaac ; Van Buren, Gene ; Nieuwenhuizen, Gerrit J. van ; Vandenbroucke, Maxence ; Varma, Raghava ; Vasconcelos, Geraldo M. S. ; Vasiliev, Alexander Nikolaevich ; Vértesi, Róbert ; Videbæk, Flemming ; Viyogi, Yogendra P. ; Vokal, Stanislav ; Voloshin, Sergei ; Vossen, A. ; Wang, J.S. ; Wang, Y. ; Wang, F. ; Wang, Y. ; Wang, G. ; Wang, H. ; Webb, Jason C. ; Webb, Grant ; Wen, L. ; Westfall, Gary D. ; Wieman, Howard ; Wissink, Scott W. ; Witt, Richard ; Wu, Y.F. ; Xiao, Z. ; Xie, W. ; Xin, K. ; Xu, Q.H. ; Xu, H. ; Xu, N. ; Xu, Y.F. ; Xu, Z. ; Yan, W. ; Yang, Y. ; Yang, Q. ; Yang, Y. ; Yang, C. ; Yang, S. ; Ye, Z. ; Yepes, Pablo P. ; Yi, L. ; Yip, K. ; Yoo, In-Kwon ; Yu, N. ; Zbroszczyk, Hanna Paulina ; Zha, W. ; Zhang, J.B. ; Zhang, X.P. ; Zhang, S. ; Zhang, Zuman ; Zhang, Y. ; Zhang, J.L. ; Zhao, F. ; Zhao, J. ; Zhong, C. ; Zhu, X. ; Zoulkarneeva, Youlia ; Zyzak, Maksym
Dihadron correlations are analyzed in √sNN = 200 GeV d + Au collisions classified by forward charged particle multiplicity and zero-degree neutral energy in the Au-beam direction. It is found that the jetlike correlated yield increases with the event multiplicity. After taking into account this dependence, the non-jet contribution on the away side is minimal, leaving little room for a back-to-back ridge in these collisions.
Adamczyk, Leszek ; Adkins, J. Kevin ; Agakishiev, Geydar ; Aggarwal, Madan Mohan ; Ahammed, Zubayer ; Alekseev, Igor G. ; Alford, J. ; Aparin, Alexey ; Arkhipkin, Dmitry A. ; Aschenauer, Elke Caroline ; Averichev, Georgy S. ; Banerjee, A. ; Bellwied, Rene ; Bhasin, Anju ; Bhati, Ashok Kumar ; Bhattarai, P. ; Bielčík, Jaroslav ; Bielčíková, Jana ; Bland, Leslie C. ; Bordyuzhin, Igor G. ; Bouchet, J. ; Brandin, Andrei V. ; Bunzarov, Ivan ; Burton, T.P. ; Butterworth, Joseph ; Caines, Helen Louise ; Calder’on de la Barca S’anchez, M. ; Campbell, J.M. ; Cebra, Daniel A. ; Cervantes, M.C. ; Chakaberia, Irakli ; Chaloupka, Petr ; Chang, Z. ; Chattopadhyay, S. ; Chen, J.H. ; Chen, X. ; Cheng, J. ; Cherney, Michael Gerard ; Christie, William ; Codrington, M.J.M. ; Contin, Giacomo ; Crawford, Henry J. ; Das, Supriya ; De Silva, L.C. ; Debbe, R.R. ; Dedovič, Tatiana G. ; Deng, J. ; Derevschikov, Anatoly A. ; di Ruzza, Benedetto ; Didenko, Lidia ; Dilks, Christopher ; Dong, X. ; Drachenberg, James Lucus ; Draper, James E. ; Du, C.M. ; Dunkelberger, L.E. ; Dunlop, James C. ; Efimov, Leonid G. ; Engelage, Jon M. ; Eppley, Geary Wareham ; Esha, Roli ; Evdokimov, Olga Y. ; Eyser, Kjeld Oleg ; Fatemi, Renee H. ; Fazio, Salvatore ; Federič, Pavol ; Fedorišin, Jan ; Feng ; Filip, Peter ; Fisyak, Yuri V. ; Flores, C.E. ; Fulek, Łukasz ; Gagliardi, Carl A. ; Garand, D. ; Geurts, Frank ; Gibson, Adam ; Girard, M. ; Greiner, Leo Clifford ; Grosnick, David P. ; Gunarathne, D.S. ; Guo, Y. ; Gupta, S. ; Gupta, Anik ; Guryn, Włodzimierz ; Hamad, Ayman ; Hamed, Ahmed M. ; Haque, R. ; Harris, John W. ; He, L. ; Heppelmann, S. ; Hirsch, Andrew S. ; Hoffmann, Gerald W. ; Hofman, D.J. ; Horvat, S. ; Huang, Huan Zhong ; Huang, X. ; Huang, Bingchu ; Huck, P. ; Humanic, Thomas J. ; Igo, George J. ; Jacobs, William W. ; Jang, H. ; Jiang, K. ; Judd, Eleanor G. ; Kabana, Sonia ; Kalinkin, Dmitry ; Kang, K. ; Kauder, Kolja ; Ke, Hongwei ; Keane, Declan ; Kechechyan, Armen ; Khan, Z.H. ; Kikola, D.P. ; Kisel, Ivan ; Kisiel, Adam Ryszard ; Klein, Spencer Robert ; Koetke, Donald D. ; Kollegger, Thorsten ; Kosarzewski, Leszek Krzysztof ; Kotchenda, L. ; Kraishan, A.F. ; Kravtsov, Peter ; Krueger, Keith William ; Kulakov, Igor ; Kumar, Lokesh ; Kycia, R.A. ; Lamont, Matthew A. C. ; Landgraf, Jeffery M. ; Landry, K.D. ; Lauret, Jerome ; Lebedev, Alexei ; Lednicky, Richard ; Lee, J.H. ; Li, X. ; Li, X. ; Li, W. ; Li, Z.M. ; Li, Y. ; Li, C. ; Lisa, Michael A. ; Liu, F. ; Ljubicic, Tonko A. ; Llope, William Joseph ; Lomnitz, M. ; Longacre, Ronald S. ; Luo, X. ; Ma, L. ; Ma, R. ; Ma, G.L. ; Ma, Yu-Gang ; Magdy Abdelwahab Abdelrahman, Niseem ; Majka, Richard Daniel ; Manion, A. ; Margetis, Spyridon ; Markert, Christina ; Masui, H. ; Matis, Howard S. ; McDonald, Daniel ; Meehan, K. ; Minaev, Nikolai G. ; Mioduszewski, Saskia ; Mohanty, Bedangadas ; Mouli, Mriganka Mouli ; Morozov, Dmitry A. ; Mustafa, M.K. ; Nandi, Basanta Kumar ; Nasim, Md. ; Nayak, Tapan Kumar ; Nigmatkulov, Grigory A. ; Nogach, Larisa V. ; Noh, S.Y. ; Novak, J. ; Nurušev, Sandibek B. ; Odyniec, Grazyna Janina ; Ogawa, Akio ; Oh, K. ; Okorokov, Vitaly A. ; Olvitt, D.L. ; Page, Brian S. ; Pan, Y.X. ; Pandit, Y. ; Panebratsev, Yuri ; Pawlak, Tomasz Jan ; Pawlik, Bogdan ; Pei, Hua ; Perkins, Chris ; Peterson, A. ; Pile, P. ; Planinic, Mirko ; Pluta, Jan Marian ; Poljak, Nikola ; Poniatowska, K. ; Porter, Jeffrey Brent ; Posik, Matthew ; Poskanzer, Arthur M. ; Pruthi, Navneet Kumar ; Putschke, Jörn H. ; Qiu, H. ; Quintero, Amilkar ; Ramachandran, Suvarna ; Raniwala, Rashmi ; Raniwala, Sudhir ; Ray, Robert L. ; Ritter, Hans Georg ; Roberts, Jabus B. ; Rogačevskij, Oleg V. ; Romero, Juan L. ; Roy, Ankhi ; Ruan, L. ; Rusnak, Jan ; Rusnakova, O. ; Sahoo, Nihar Ranjan ; Sahu, Pradip Kumar ; Sakrejda, Iwona ; Salur, Sevil ; Sandacz, A. ; Sandweiss, Jack H. ; Sarkar, Amal ; Schambach, Joachim ; Scharenberg, Rolf Paul ; Schmah, Alexander ; Schmidke, William B. ; Schmitz, Norbert ; Seger, Janet Elizabeth ; Seyboth, Peter ; Shah, N. ; Shahaliev, Ehtiram ; Shanmuganathan, Prashanth V. ; Shao, M. ; Sharma, M.K. ; Sharma, B. ; Shen, W.Q. ; Shi, Shusu ; Shou, Q.Y. ; Sichtermann, Ernst P. ; Sikora, Rafał ; Šimko, Miroslav ; Skoby, Michael J. ; Smirnov, Nikolai ; Smirnov, Dmitri V. ; Solanki, D. ; Song, L. ; Sorensen, Paul Richard ; Spinka, Harold. 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The acceptance-corrected dielectron excess mass spectra, where the known hadronic sources have been subtracted from the inclusive dielectron mass spectra, are reported for the first time at mid-rapidity |yee|<1 in minimum-bias Au+Au collisions at sNN−−−−√ = 19.6 and 200 GeV. The excess mass spectra are consistently described by a model calculation with a broadened ρ spectral function for Mee<1.1 GeV/c2. The integrated dielectron excess yield at sNN−−−−√ = 19.6 GeV for 0.4<Mee<0.75 GeV/c2, normalized to the charged particle multiplicity at mid-rapidity, has a value similar to that in In+In collisions at sNN−−−−√ = 17.3 GeV. For sNN−−−−√ = 200 GeV, the normalized excess yield in central collisions is higher than that at sNN−−−−√ = 17.3 GeV and increases from peripheral to central collisions. These measurements indicate that the lifetime of the hot, dense medium created in central Au+Au collisions at sNN−−−−√ = 200 GeV is longer than those in peripheral collisions and at lower energies.