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Institute
Die Reichsstelle für den Unterrichtsfilm (später Reichsanstalt für Film und Bild in Wissenschaft und Unterricht ) stellte - wie ihr Name sagt - den Unterrichtsfilm in den Mittelpunkt ihrer Arbeit. Das Lichtbild wurde zwar schon im Einführungserlaß des Reichserziehungsministeriums vom 26. Juni 1934 mehrfach erwähnt, trat aber - wie auch die Schallplatte - erst später hervor. ...
Muthukumar, Yazh ; Münkemer, Johanna ; Mathieu, Daniel ; Richter, Christian ; Schwalbe, Harald ; Steinmetz, Heinrich ; Kessler, Wolfgang ; Reichelt, Joachim ; Beutling, Ulrike ; Frank, Ronald ; Büssow, Konrad ; Heuvel, Joop van den ; Brönstrup, Mark ; Taylor, Richard E. ; Laschat, Sabine ; Sasse, Florenz
The identification of inhibitors of eukaryotic protein biosynthesis, which are targeting single translation factors, is highly demanded. Here we report on a small molecule inhibitor, gephyronic acid, isolated from the myxobacterium Archangium gephyra that inhibits growth of transformed mammalian cell lines in the nM range. In direct comparison, primary human fibroblasts were shown to be less sensitive to toxic effects of gephyronic acid than cancer-derived cells. Gephyronic acid is targeting the protein translation system. Experiments with IRES dual luciferase reporter assays identified it as an inhibitor of the translation initiation. DARTs approaches, co-localization studies and pull-down assays indicate that the binding partner could be the eukaryotic initiation factor 2 subunit alpha (eIF2α). Gephyronic acid seems to have a different mode of action than the structurally related polyketides tedanolide, myriaporone, and pederin and is a valuable tool for investigating the eukaryotic translation system. Because cancer derived cells were found to be especially sensitive, gephyronic acid could potentially find use as a drug candidate.
Molnar, Wolfgang ; Lugstein, Alois ; Wojcik, Tomasz ; Pongratz, Peter ; Auner, Norbert ; Bauch, Christian ; Bertagnolli, Emmerich
Perchlorinated polysilanes were synthesized by polymerization of tetrachlorosilane under cold plasma conditions with hydrogen as a reducing agent. Subsequent selective cleavage of the resulting polymer yielded oligochlorosilanes SinCl2n+2 (n = 2, 3) from which the octachlorotrisilane (n = 3, Cl8Si3, OCTS) was used as a novel precursor for the synthesis of single-crystalline Si nanowires (NW) by the well-established vapor–liquid–solid (VLS) mechanism. By adding doping agents, specifically BBr3 and PCl3, we achieved highly p- and n-type doped Si-NWs by means of atmospheric-pressure chemical vapor deposition (APCVD). These as grown NWs were investigated by means of scanning electron microscopy (SEM) and transmission electron microscopy (TEM), as well as electrical measurements of the NWs integrated in four-terminal and back-gated MOSFET modules. The intrinsic NWs appeared to be highly crystalline, with a preferred growth direction of [111] and a specific resistivity of ρ = 6 kΩ·cm. The doped NWs appeared to be [112] oriented with a specific resistivity of ρ = 198 mΩ·cm for p-type Si-NWs and ρ = 2.7 mΩ·cm for n-doped Si-NWs, revealing excellent dopant activation.
From 12.12.2010 to 17.12.2010, the Dagstuhl Seminar 10501 "Advances and Applications of Automata on Words and Trees" was held in Schloss Dagstuhl - Leibniz Center for Informatics. During the seminar, several participants presented their current research, and ongoing work and open problems were discussed. Abstracts of the presentations given during the seminar as well as abstracts of seminar results and ideas are put together in this paper. The first section describes the seminar topics and goals in general. Links to extended abstracts or full papers are provided, if available.
Seminar: 10501 - Advances and Applications of Automata on Words and Trees. The aim of the seminar was to discuss and systematize the recent fast progress in automata theory and to identify important directions for future research. For this, the seminar brought together more than 40 researchers from automata theory and related fields of applications. We had 19 talks of 30 minutes and 5 one-hour lectures leaving ample room for discussions. In the following we describe the topics in more detail.
Seit Dezember 2003 warteten viele Arachnologen auf eine Aktualisierung des Internetbestimmungsschlüssels „Spinnen Mitteleuropas“. Die Umstellung des Systems von html auf php erwies sich aufgrund des komplexen Themas als umfangreicher als gedacht. Mit Daniel Gloor haben wir nun einen Datenbankund Internet-Fachmann in unseren Reihen, der sich (auch) dieser technischen Probleme annimmt.
Thamm, Markus ; Rolke, Daniel ; Jordan, Nadine ; Balfanz, Sabine ; Schiffer, Christian ; Baumann, Arnd ; Blenau, Wolfgang
Background: Serotonin plays a pivotal role in regulating and modulating physiological and behavioral processes in both vertebrates and invertebrates. In the honeybee (Apis mellifera), serotonin has been implicated in division of labor, visual processing, and learning processes. Here, we present the cloning, heterologous expression, and detailed functional and pharmacological characterization of two honeybee 5-HT2 receptors.
Methods: Honeybee 5-HT2 receptor cDNAs were amplified from brain cDNA. Recombinant cell lines were established constitutively expressing receptor variants. Pharmacological properties of the receptors were investigated by Ca2+ imaging experiments. Quantitative PCR was applied to explore the expression patterns of receptor mRNAs.
Results: The honeybee 5-HT2 receptor class consists of two subtypes, Am5-HT2α and Am5-HT2β. Each receptor gene also gives rise to alternatively spliced mRNAs that possibly code for truncated receptors. Only activation of the full-length receptors with serotonin caused an increase in the intracellular Ca2+ concentration. The effect was mimicked by the agonists 5-methoxytryptamine and 8-OH-DPAT at low micromolar concentrations. Receptor activities were blocked by established 5-HT receptor antagonists such as clozapine, methiothepin, or mianserin. High transcript numbers were detected in exocrine glands suggesting that 5-HT2 receptors participate in secretory processes in the honeybee.
Conclusions: This study marks the first molecular and pharmacological characterization of two 5-HT2 receptor subtypes in the same insect species. The results presented should facilitate further attempts to unravel central and peripheral effects of serotonin mediated by these receptors.
Frölich, Lutz ; Peters, Oliver ; Lewczuk, Piotr ; Gruber, Oliver ; Teipel, Stefan ; Gertz, Hermann-Josef ; Jahn, Holger ; Jessen, Frank ; Kurz, Alexander ; Luckhaus, Christian ; Hüll, Michael ; Pantel, Johannes ; Reischies, Friedel ; Schröder, Johannes ; Wagner, Michael ; Rienhoff, Otto ; Wolf, Stefanie ; Bauer, Chris ; Schuchhardt, Johannes ; Heuser, Isabella ; Rüther, Eckart ; Henn, Fritz ; Maier, Wolfgang ; Wiltfang, Jens ; Kornhuber, Johannes
Background: The progression of mild cognitive impairment (MCI) to Alzheimer’s disease (AD) dementia can be predicted by cognitive, neuroimaging, and cerebrospinal fluid (CSF) markers. Since most biomarkers reveal complementary information, a combination of biomarkers may increase the predictive power. We investigated which combination of the Mini-Mental State Examination (MMSE), Clinical Dementia Rating (CDR)-sum-of-boxes, the word list delayed free recall from the Consortium to Establish a Registry of Dementia (CERAD) test battery, hippocampal volume (HCV), amyloid-beta1–42 (Aβ42), amyloid-beta1–40 (Aβ40) levels, the ratio of Aβ42/Aβ40, phosphorylated tau, and total tau (t-Tau) levels in the CSF best predicted a short-term conversion from MCI to AD dementia.
Methods: We used 115 complete datasets from MCI patients of the "Dementia Competence Network", a German multicenter cohort study with annual follow-up up to 3 years. MCI was broadly defined to include amnestic and nonamnestic syndromes. Variables known to predict progression in MCI patients were selected a priori. Nine individual predictors were compared by receiver operating characteristic (ROC) curve analysis. ROC curves of the five best two-, three-, and four-parameter combinations were analyzed for significant superiority by a bootstrapping wrapper around a support vector machine with linear kernel. The incremental value of combinations was tested for statistical significance by comparing the specificities of the different classifiers at a given sensitivity of 85%.
Results: Out of 115 subjects, 28 (24.3%) with MCI progressed to AD dementia within a mean follow-up period of 25.5 months. At baseline, MCI-AD patients were no different from stable MCI in age and gender distribution, but had lower educational attainment. All single biomarkers were significantly different between the two groups at baseline. ROC curves of the individual predictors gave areas under the curve (AUC) between 0.66 and 0.77, and all single predictors were statistically superior to Aβ40. The AUC of the two-parameter combinations ranged from 0.77 to 0.81. The three-parameter combinations ranged from AUC 0.80–0.83, and the four-parameter combination from AUC 0.81–0.82. None of the predictor combinations was significantly superior to the two best single predictors (HCV and t-Tau). When maximizing the AUC differences by fixing sensitivity at 85%, the two- to four-parameter combinations were superior to HCV alone.
Conclusion: A combination of two biomarkers of neurodegeneration (e.g., HCV and t-Tau) is not superior over the single parameters in identifying patients with MCI who are most likely to progress to AD dementia, although there is a gradual increase in the statistical measures across increasing biomarker combinations. This may have implications for clinical diagnosis and for selecting subjects for participation in clinical trials.
Berufliche Qualifikationsmismatches bei Zugängen in Arbeitslosigkeit : ein Diskussionsbeitrag
(2013)
Baden, Christian ; Gericke, Pierre-Andre ; Hasberg, Ruth ; Klems, Wolfgang ; Schmid, Alfons ; Werth, Stefan
Die Bedeutung von Diskrepanzen zwischen den Qualifikationen und Fähigkeiten der Erwerbstätigen und den Jobanforderungen für die wirtschaftliche Entwicklung und Wettbewerbsfähigkeit wird vor allem international in jüngster Zeit zunehmend diskutiert und thematisiert. Die Gründe dafür liegen u.a. darin, dass sich bei solchen Diskrepanzen die Arbeitszufriedenheit und die Produktivität in Betrieben verringern und es zu einem Verlust von Humankapital und zur Reduktion des Produktivitätswachstums kommt.
In Deutschland ist diese Diskussion zumindest auf wirtschafts- und arbeitsmarktpolitischer Ebene bisher eher von zweitrangiger Bedeutung. Dieser Beitrag richtet sich entsprechend auf die
Beantwortung der Frage, welches Ausmaß der berufliche
Qualifikationsmismatch in der Bundesrepublik Deutschland hat. Aufgrund der (noch) bestehenden Datensituation werden Mismatches bei den Qualifikationen für die Zugänge von Personen in Arbeitslosigkeit untersucht. Diese Begrenzung hat primär datentechnische Gründe, für die Beschäftigten liegen die Daten noch nicht vor. Mismatches bei Zugängen in Arbeitslosigkeit sind aber auch wissenschaftlich von Interesse, da u.W. bisher keine systematische Analyse dafür erfolgte.
Die empirische Untersuchung über Qualifikationsmismatches bei Zugängen in Arbeitslosigkeit wird nach verschiedenen Kategorien ausdifferenziert. So interessieren mögliche Unterschiede nach Geschlecht, Alter und schwerpunktmäßig nach (ausgewählten) Berufen bzw. Berufsgruppen. Als Datenbasis dient die Arbeitslosenstatistik der BA. Diese hat den Vorteil, dass die formalen Bildungsabschlüsse arbeitslos gewordener Personen den geforderten Qualifikationen ihrer vorangegangenen Beschäftigung gegenübergestellt werden können. Zudem lassen sich mit dieser Statistik unterschiedliche Berufe und Personengruppen detailliert untersuchen.
Für die Zugänge in Arbeitslosigkeit lässt sich nach den Untersuchungsergebnissen konstatieren, dass formale Qualifikation und Anforderungsniveau weitgehend übereinstimmen. Allerdings gab es
bei den Zugängen in Arbeitslosigkeit immerhin bei knapp 30% eine
Diskrepanz zwischen Ausbildung und der zuletzt ausgeübter Tätigkeit. Der Anteil an Personen, deren formale unterhalb der geforderten Qualifikation lag (Unterqualifizierung/überwertige Beschäftigung), war etwas größer als der Anteil der Personen mit einem höheren als dem geforderten Qualifikationsniveau Überqualifizierung/unterwertige Beschäftigung).
Die Differenzierung nach einigen ausgewählten Kriterien ergab keine größeren Unterschiede bei der Passung wie auch bei den Mismatches. Weder bestanden größere Abweichungen zwischen den Bundesländern noch gab es gravierende Unterschiede nach dem Geschlecht, dem Alter und nach Qualifikationsklassen und Anforderungsniveaus. Auf diese Strukturfaktoren lassen sich die konstatierten Mismatches somit nicht zurückführen.
Bei den untersuchten Berufen lässt sich resümierend als erstes festhalten, dass bei allen Personen, die sich im Untersuchungszeitraum arbeitslos gemeldet haben, die passgenaue Beschäftigung, gemessen am Ausbildungsberuf und an den Anforderungsniveaus der Tätigkeit, die die Personen ausübten, bei weitem überwog; allerdings schwankten die Anteile bei der Übereinstimmung zwischen 56% bei den Lagerverwaltern/Magazinern und 83% bei den Malern/Lackieren. Entsprechend lässt sich zum zweiten konstatieren, dass in allen Berufen Mismatches hinsichtlich unterqualifizierter (überwertiger) und überqualifizierter (unterwertiger) Beschäftigung in der vorherigen Beschäftigung bestanden, diese aber unterschiedlich hoch in den einzelnen Berufen waren.
Die untersuchten Berufsaggregate und die zehn Berufe lassen sich grob in drei Kategorien bezüglich der Mismatches einteilen. Bei einigen Berufen überwiegt die überqualifizierte Beschäftigung, d.h. die sich arbeitslos Meldenden waren in ihrer vorherigen Tätigkeit unter ihrer formalen Qualifikation beschäftigt. Bei den Berufsaggregaten waren das Grüne Berufe und Gesundheitsberufe; bei den Berufen: Lagerverwalter/Magaziner, Maler/Lackierer und Maurer, wobei der Anteil der Überqualifikation variierte. In etwa gleich hoch sind die Anteile der über- und unterqualifizierten Beschäftigung bei Köchen, Bürofachkräften und Verkäufer/innen. Bei den übrigen Berufen überwiegt eine unterqualifizierte Beschäftigung vor der Meldung in Arbeitslosigkeit: Transport- und Logistik, wissensintensive Berufe, MINT-Berufe sowie Kellner/Stewards, Kraftfahrzeugführer, Groß- und Einzelhandelskaufleute/ Einkäufer.
Was die Ursachen für diese Unterschiede sind, lässt sich nach den vorliegenden Ergebnissen nicht beantworten. Ein Teil der Diskrepanzen dürfte, wie bereits erwähnt, auf die Qualifikationsniveaus der Berufe selbst zurückzuführen sein. Allerdings trägt auch dieser Erklärungsversuch nur teilweise. Dies verdeutlicht der Beruf Einzelhandelskaufleute. Trotz eines im Durchschnitt mittleren Anforderungsniveaus bei dieser Berufsgruppe, findet man dort Personen mit abgeschlossener Berufsausbildung, die überwiegend sogar zwei Qualifikationsstufen höher arbeiteten.
Insgesamt lässt sich festhalten, dass hinsichtlich der Erklärung von über- und unterwertiger Beschäftigung bei Zugängen in Arbeitslosigkeit noch einiger Forschungsbedarf besteht
Hinz, Oliver ; Pfeuffer, Nicolas ; Stammer, Wolfgang ; Schramowski, Patrick ; Abdel-Karim, Benjamin M. ; Bucher, Andreas ; Hügel, Christian ; Rohde, Gernot Gerhard Ulrich ; Kersting, Kristian
COVID-19 HAS AGAIN TIGHTENED ITS GRIP AROUND THE WORLD AND THE HEALTH SYSTEM. THIS ARTICLE GIVES AN INTRODUCTION TO EXPLAINABLE INTERACTIVE MACHINE LEARNING AND PROVIDES INSIGHTS ON HOW THIS METHOD MAY NOT ONLY HELP IN ENGINEERING MORE POWERFUL AI SYSTEMS, BUT ALSO HOW IT MAY HELP TO EASE THE BURDEN OF VIRAL STRAINS ON THE HEALTHCARE SYSTEM.