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We adopt Markert and Nissim (2005)’s approach of using the World Wide Web to resolve cases of coreferent bridging for German and discuss the strength and weaknesses of this approach. As the general approach of using surface patterns to get information on ontological relations between lexical items has only been tried on English, it is also interesting to see whether the approach works for German as well as it does for English and what differences between these languages need to be accounted for. We also present a novel approach for combining several patterns that yields an ensemble that outperforms the best-performing single patterns in terms of both precision and recall.
Prieto García, Cristian ; Hartmann, Oliver ; Reissland, Michaela ; Braun, Fabian ; Bozkurt, Süleyman ; Fuß, Carmina Teresa ; Schülein-Völk, Christina ; Buchberger, Alexander ; Calzado Canale, Marco A. ; Rosenfeldt, Mathias Tillmann ; Đikić, Ivan ; Münch, Christian ; Diefenbacher, Markus Elmar
Oncogenic transformation of lung epithelial cells is a multi-step process, frequently starting with the inactivation of tumor suppressors and subsequent activating mutations in proto-oncogenes, such as members of the PI3K or MAPK family. Cells undergoing transformation have to adjust to changes, such as metabolic requirements. This is achieved, in part, by modulating the protein abundance of transcription factors, which manifest these adjustments. Here, we report that the deubiquitylase USP28 enables oncogenic reprogramming by regulating the protein abundance of proto-oncogenes, such as c-JUN, c-MYC, NOTCH and ΔNP63, at early stages of malignant transformation. USP28 is increased in cancer compared to normal cells due to a feed-forward loop, driven by increased amounts of oncogenic transcription factors, such as c-MYC and c-JUN. Irrespective of oncogenic driver, interference with USP28 abundance or activity suppresses growth and survival of transformed lung cells. Furthermore, inhibition of USP28 via a small molecule inhibitor reset the proteome of transformed cells towards a ‘pre-malignant’ state, and its inhibition cooperated with clinically established compounds used to target EGFRL858R, BRAFV600E or PI3KH1047R driven tumor cells. Targeting USP28 protein abundance already at an early stage via inhibition of its activity therefore is a feasible strategy for the treatment of early stage lung tumours and the observed synergism with current standard of care inhibitors holds the potential for improved targeting of established tumors.
Voskamp, Alke ; Fritz, Susanne A. ; Köcke, Anna Valerie ; Biber, Matthias ; Nogueira-Brockmeyer, Timo ; Bertzky, Bastian ; Forrest, Matthew ; Goldstein, Allie ; Henderson, Scott ; Hickler, Thomas ; Hof, Christian ; Kastner, Thomas ; Lang, Stefanie ; Manning, Peter ; Mascia, Michael B. ; McFadden, Ian R. ; Niamir, Aidin ; Noon, Monica ; O’Donell, Brian ; Opel, Mark ; Schwede, Georg ; West, Peyton ; Schenck, Christof ; Böhning-Gaese, Katrin
The establishment and maintenance of protected areas (PAs) is viewed as a key action in delivering post-2020 biodiversity targets. PAs often need to meet multiple objectives, ranging from biodiversity protection to ecosystem service provision and climate change mitigation, but available land and conservation funding is limited. Therefore, optimizing resources by selecting the most beneficial PAs is vital. Here, we advocate for a flexible and transparent approach to selecting protected areas based on multiple objectives, and illustrate this with a decision support tool on a global scale. The tool allows weighting and prioritization of different conservation objectives according to user-specified preferences, as well as real-time comparison of the selected areas that result from such different priorities. We apply the tool across 1347 terrestrial PAs and highlight frequent trade-offs among different objectives, e.g., between species protection and ecosystem integrity. Outputs indicate that decision makers frequently face trade-offs among conflicting objectives. Nevertheless, we show that transparent decision-support tools can reveal synergies and trade-offs associated with PA selection, thereby helping to illuminate and resolve land-use conflicts embedded in divergent societal and political demands and values.
In this paper, we argue that difficulties in the definition of coreference itself contribute to lower inter-annotator agreement in certain cases. Data from a large referentially annotated corpus serves to corroborate this point, using a quantitative investigation to assess which effects or problems are likely to be the most prominent. Several examples where such problems occur are discussed in more detail, and we then propose a generalisation of Poesio, Reyle and Stevenson’s Justified Sloppiness Hypothesis to provide a unified model for these cases of disagreement and argue that a deeper understanding of the phenomena involved allows to tackle problematic cases in a more principled fashion than would be possible using only pre-theoretic intuitions.
Fedchenko, Olena ; Song, Young-Joon ; Tkač, Olena ; Lytvynenko, Yaryna ; Chernov, Sergii ; Gloskovskii, Andrei ; Schlueter, Christoph ; Peters, Marius ; Kliemt, Kristin ; Krellner, Cornelius ; Valentí, Roser ; Schönhense, Gerd ; Elmers, Hans-Joachim
We present results of hard X-ray angle-resolved photoemission spectroscopy and photoemission diffraction measurements performed on high-quality single crystals of the valence transition compound EuPd2Si2 for temperatures 25~K ≤ T ≤ 300~K. At low temperatures we observe a Eu 4f valence v=2.5, % occupation number n=6.5, which decreases to v=2.1 for temperatures above the valence transition around TV≈160~K. The experimental valence numbers resulting from an evaluation of the Eu(III)/Eu(II) 3d core levels, are used for calculating band structures using density functional theory. The valence transition significantly changes the band structure as determined by angle-resolved photoemission spectroscopy. In particular, the Eu 5d valence bands are shifted to lower binding energies with increasing Eu 4f occupancy. To a lesser extent, bands derived from the Si 3p and Pd 4d orbitals are also affected. This observation suggests a partial charge transfer between Eu and Pd/Si sites. Comparison with {\it ab-initio} theory shows a good agreement with experiment, in particular concerning the unequal band shift with increasing Eu 4f occupancy.
Conventional cluster and virial expansions are generalized to momentum dependent interparticle potentials. The model with Lorentz contracted hard core potentials is considered, e.g. as hadron gas model. A Van der Waals-type model with a temperature dependent excluded volume is derived. Lorentz contraction effects at given temperature are stronger for light particles and make their effective excluded volume smaller than that of heavy ones.
Sprachwahl und Sprachwahrnehmung sind im Deutschen unabdingbar geprägt durch das Wissen von einer Standardsprache. Dieses Wissen basiert für die meisten Sprecher auf der Erfahrung, dass in der Schule manche sprachliche Formen als korrekt, andere als falsch bewertet werden, außerdem auf der Tatsache, dass es Fixierungen der Regeln des Standards in Lexika und Grammatiken gibt. Wissen und Anerkennung dieses Standards sind unabhängig davon, dass keine dieser Kodifikationen unumstritten ist, dass viele Sprecher die Regeln nicht genau kennen und dass als Vorbilder anerkannte Personen (Nachrichtensprecher, Journalisten bestimmter Zeitschriften, Lehrer, Literaten u.a.) keineswegs einheitliche Regeln verfolgen. Der Standard ist fest assoziiert mit der Erfahrung einer legitimen Regelhaftigkeit, also mit Ordnung. Verwendung von Nonstandard wird mit Bezug auf diese Ordnung und von ihr unterschieden wahrgenommen. Diese relationale Sicht der Dinge ist sowohl subjektiv als auch intersubjektiv.
In der deutschsprachigen Schweiz stehen sich gesprochene Mundarten und geschriebene Standardsprache gegenüber. Außer in formellen Situationen wird Mundart gesprochen, und bis vor kurzem wurde nur selten Mundart geschrieben, sondern die hochdeutsche Schriftsprache. Die Chat-Kommunikation zeigt einerseits durch die nicht-zeitversetzte quasi-direkte Kommunikation wesentliche Züge von Mündlichkeit, die zusammen mit der Informalität im Chat den Mundartgebrauch fördert. Andererseits ist das Medium immer noch die Schrift, welche die Domäne der Standardsprache darstellt. Mundart und Standardsprache stehen sich also in Chaträumen in direkter Konkurrenz gegenüber. Der folgende Beitrag analysiert quantitativ und qualitativ das Neben- und Miteinander der beiden Varietäten in Schweizer Chaträumen und untersucht das Vorkommen und die Bedingungen von Code-Alternation und Code-Switches.
Winter, Andreas ; Nepper, Pascal ; Hermann, Marcus ; Bayer, Franziska ; Rieß, Stephanie ; Marinos, Spiros Lukas ; Linden, Arnaud van ; Holubec, Tomas ; Steinbicker, Andrea U. ; Zacharowski, Kai ; Walther, Thomas ; Emrich, Fabian Christoph
Background Vasoplegic syndrome is frequently observed during cardiac surgery and resembles a complication of high mortality and morbidity. There is a clinical need for therapy and prevention of vasoplegic syndrome during complex cardiac surgical procedures. Therefore, we investigated different strategies in a porcine model of vasoplegia.
Methods We evaluated new medical therapies and prophylaxis to avoid vasoplegic syndrome in a porcine model. After induction of anesthesia, cardiopulmonary bypass was established through median sternotomy and central cannulation. Prolonged aortic cross-clamping (120 min) simulated a complex surgical procedure. The influence of sevoflurane-guided anesthesia (sevoflurane group) and the administration of glibenclamide (glibenclamide group) were compared to a control group, which received standard anesthesia using propofol. Online hemodynamic assessment was performed using PiCCO® measurements. In addition, blood and tissue samples were taken to evaluate hemodynamic effects and the degree of inflammatory response.
Results Glibenclamide was able to break through early vasoplegic syndrome by raising the blood pressure and systemic vascular resistance as well as less need of norepinephrine doses. Sevoflurane reduced the occurrence of the vasoplegic syndrome in the mean of stable blood pressure and less need of norepinephrine doses.
Conclusion Glibenclamide could serve as a potent drug to reduce effects of vasoplegic syndrome. Sevoflurane anesthesia during cardiopulmonary bypass shows less occurrence of vasoplegic syndrome and therefore could be used to prevent it in high-risk patients.
Clinical Perspective; what is new?
* to our knowledge, this is the first randomized in vivo study evaluating the hemodynamic effects of glibenclamide after the onset of vasoplegic syndrome
* furthermore according to literature research, there is no study showing the effect of sevoflurane-guided anesthesia on the occurrence of a vasoplegic syndrome
Clinical Perspective; clinical implications?
to achieve better outcomes after complex cardiac surgery there is a need for optimized drug therapy and prevention of the vasoplegic syndrome